Natural Product Synthesis & Reaction Discovery

Garg Research Group

 

Independent Career


89. Understanding and Interrupting the Fischer Azaindolization Reaction.

      Bryan J. Simmons, Marie Hoffmann, Pier Alexandre Champagne, Elias Picazo, Katsuya Yamakawa, Lucas A. Morrill, K. N. Houk, and Neil K.
      Garg. J. Am. Chem. Soc. 2017, Article ASAP.

     Abstract | PDF | Supporting Information




88. Engineering the Biocatalytic Selectivity of Iridoid Production in Saccharomyces cerevisiae.

      John M. Billingsley, Anthony B. DeNicola, Joyann S. Barber, Man-Cheng Tang, Joe Horecka, Angela Chu, Neil K. Garg, and Yi Tang.
      Metab. Eng. 2017, 44, 117–125.

     Abstract | PDF | Supporting Information



  1. 87.Spectroscopy 101: A Practical Introduction to Spectroscopy and Analysis for Undergraduate Organic Chemistry Laboratories.

      Lucas A. Morrill, Jacquelin K. Kammeyer, and Neil. K. Garg. J. Chem. Educ. 2017, Article ASAP.

     Abstract | PDF | Supporting Information




  1. 86.Conjugated Trimeric Scaffolds Accessible from Indolyne Cyclotrimerizations: Synthesis, Structures, and Electronic Properties.

      Janice B. Lin, Tejas K. Shah, Adam E. Goetz, Neil K. Garg, and K. N. Houk. J. Am. Chem. Soc. 2017, 139, 10447–10455.

      Abstract | PDF | Supporting Information | Synfacts Highlight




85. Indole Diterpenoid Natural Products as the Inspiration for New Synthetic Methods and Strategies.

      Michael A. Corsello, Junyong Kim, and Neil K. Garg. Chem. Sci. 2017, 8, 5836–5844.

      Abstract | PDF




84. Total Synthesis of ()-Tubingensin B Enabled by the Strategic Use of an Aryne Cyclization.

      Michael A. Corsello, Junyong Kim, and Neil K. Garg. Nat. Chem. 2017, 9, 944–949.

      Abstract | PDF | Supporting Information | Synfacts Highlight
































83. Enantioselective Nickel-Catalyzed Mizoroki–Heck Cyclizations to Generate Quaternary Stereocenters.

     Jean-Nicolas Desrosiers, Jialin Wen, Sergei Tcyrulnikov, Soumik Biswas, Bo Qu, Liana Hie, Dmitry Kurouski, Ling Wu, Nelu Grinberg, Nizar

     Haddad, Carl A. Busacca, Nathan K. Yee, Jinhua J. Song, Neil K. Garg, Xumu Zhang, Marisa C. Kozlowski, and Chris H. Senanayake.

     Org. Lett. 2017, 19, 3338–3341.

     Abstract | PDF | Supporting Information




82. Kinetic Modeling of the Nickel-Catalyzed Esterification of Amides.

       Nicholas A. Weires, Daniel D. Caspi, and Neil K. Garg. ACS Catal. 2017, 7, 4381–4385.

     Abstract | PDF | Supporting Information | ACS Editor’s Choice (June 4, 2017) | C&E News



81. Mizoroki–Heck Cyclizations of Amide Derivatives for the Introduction of Quaternary Centers.

       Jose M. Medina, Jesus Moreno, Sophie Racine, Shuaijing Du, and Neil K. Garg. Angew. Chem., Int. Ed. 2017, 56, 6567–6571.

     Abstract | PDF | Supporting Information




  1. 80.The Organic Coloring Book.

      Elaina Garg, Kaylie Garg, and Neil K. Garg.

      Available at Amazon | C&E News




79. Collaborative Biosynthesis of Maleimide- and Succinimide-Containing Natural Products by Fungal Polyketide Megasynthases.

      Michio Sato, Jacob E. Dander, Chizuru Sato, Yiu-sun Hung, Shu-Shan Gao, Man-Cheng Tang, Leibniz Hang, Jaclyn M. Winter, Neil K. Garg,
      Kenji Watanabe, and Yi Tang
. J. Am. Chem. Soc. 2017, 139, 53175320.

      Abstract | PDF | Supporting Information



78. Nickel-Catalyzed Reduction of Secondary and Tertiary Amides.

      Bryan J. Simmons, Marie Hoffmann, Jaeyeon Hwang, Moritz K. Jackl, and Neil K. Garg. Org. Lett. 2017, 19, 1910–1913.

      Abstract | PDF | Supporting Information



77. Enzyme-Catalyzed Stereoselective Intramolecular Hydroalkoxylation.

      Shu-Shan Gao, Marc Garcia-Borràs, Joyann S. Barber, Yang Hai, Abing Duan, Neil K. Garg, K. N. Houk, and Yi Tang. J. Am. Chem. Soc.
     
2017, 139, 36393642.

      Abstract | PDF | Supporting Information | SYNFACTS Highlights




76. Organic Chemistry Can Sizzle.

      Tejas K. Shah, and Neil K. Garg. Nat. Rev. Chem. 2017, 1, 1–3.

      Abstract | PDF


75. Breaking Amides Using Nickel Catalysis.

      Jacob E. Dander and Neil K. Garg. ACS Catal. 2017, 7, 1413–1423.

      Abstract | PDF




  1. 74.Expanding the ROMP Toolbox: Synthesis of Air-Stable Benzonorbornadiene Polymers by Aryne Chemistry.

      Jose M. Medina, Jeong Hoon Ko, Heather D. Maynard, and Neil K. Garg. Macromolecules 2017, 50, 580–586.

      Abstract | PDF | Supporting Information




  1. 73.Pardon the Interruption: A Modification of Fischer’s Venerable ­Reaction for the Synthesis of Heterocycles and Natural Products.

      Robert B. Susick, Lucas A. Morrill, Elias Picazo, and Neil K. Garg. Synlett 2017, 28, 1–11.

      Abstract | PDF




72. Nickel-Catalyzed Esterification of Aliphatic Amides.

      Liana Hie, Emma L. Baker, Sarah M. Anthony, Jean-Nicolas Desrosiers, Chris Senanayake, and Neil K. Garg.
      Angew. Chem. Int. Ed. 2016, 55, 15129–15132.

      Abstract | PDF | Supporting Information




71. Nickel-Catalyzed Suzuki-Miyaura Coupling in t-Amyl Alcohol for the Preparation of 5-(Furan-3-yl)pyrimidine.

      Liana Hie and Neil K. Garg. Org. Synth. 2016, 93, 306–318.

      Abstract | PDF




  1. 70.Quantification of the Electrophilicity of Benzyne and Related Intermediates.

      Noah F. Fine Nathel, Lucas A. Morrill, Herbert Mayr, and Neil K. Garg. J. Am. Chem. Soc. 2016, 138, 10402–10405.

      Abstract | PDF | Supporting Information




  1. 69.Construction of Quaternary Stereocenters via Nickel-Catalyzed Heck Cyclizations.

      Jean-Nicolas Desrosiers, Liana Hie, Soumik Biswas, Olga V. Zatolochnaya, Sonia Rodriguez, Heewon Lee, Nelu Grinberg, Nizar Haddad,

      Nathan K. Yee, Neil K. Garg, and Chris H. Senanayake.

      Angew. Chem. Int. Ed. 2016, 55, 11921–11924.

      Abstract | PDF | Supporting Information




  1. 68.Benchtop Delivery of Ni(cod)2 using Paraffin Capsules.

      Jacob E. Dander, Nicholas A. Weires, and Neil K. Garg. Org. Lett. 2016, 18, 3934–3936.

      Abstract | PDF | Supporting Information




67. A Two-Step Approach to Achieve Secondary Amide Transamidation Enabled by Nickel Catalysis.

      Emma L. Baker, Michael M. Yamano, Yujing Zhou, Sarah M. Anthony, and Neil K. Garg. Nat. Commun. 2016, 7, 1–5.

      Abstract | PDF | Supporting Information




  1. 66.Nickel-Catalyzed Alkylation of Amide Derivatives.

      Bryan J. Simmons, Nicholas A. Weires, Jacob E. Dander, and Neil K. Garg. ACS Catal. 2016, 6, 3176–3179.

      Abstract | PDF | Supporting Information




65. Expanding the Strained Alkyne Toolbox: Generation and Utility of Oxygen-Containing Strained Alkynes.

        Tejas K. Shah, Jose M. Medina, and Neil K. Garg. J. Am. Chem. Soc. 2016, 138, 4948–4954.

      Abstract | PDF | Supporting Information




64. P450-Mediated Coupling of Indole Fragments to Forge Communesin and Unnatural Isomers.

      Hsiao-Ching Lin, Travis C. McMahon, Ashay Patel, Michael Corsello, Adam Simon, Wei Xu, Muxun Zhao, K. N. Houk, Neil K. Garg,

      and Yi Tang. J. Am. Chem. Soc. 2016, 138, 4002–4005.

        Abstract | PDF | Supporting Information




  1. 63.Synthetic Studies Pertaining to the 2,3-Pyridyne and 4,5-Pyrimidyne.
    Jose M. Medina, Moritz K. Jackl, Robert B. Susick, and Neil K. Garg. Tetrahedron 2016, 72, 3629–3634.

      Abstract | PDF | Supporting Information




  1. 62.Nitrone Cycloadditions of 1,2-Cyclohexadiene.
    Joyann S. Barber, Evan D. Styduhar, Hung V. Pham, Travis C. McMahon, K. N. Houk, and Neil K. Garg.

      J. Am. Chem. Soc. 2016, 138, 2512–2515.

      Abstract | PDF | Supporting Information

     


61. Enantioselective Total Syntheses of Akuammiline Alkaloids (+)-Strictamine, (–)-2(S)-Cathafoline, and (–)-Aspidophylline A.

      Jesus Moreno, Elias Picazo, Lucas A. Morrill, Joel M. Smith, and Neil K. Garg. J. Am. Chem. Soc. 2016, 138, 1162–1165.

      Abstract | PDF | Supporting Information




  1. 60.Nickel-Catalyzed Activation of Acyl C–O Bonds of Methyl Esters.

      Liana Hie, Noah F. Fine Nathel, Xin Hong, Yun-Fang Yang, K. N. Houk, and Neil K. Garg. Angew. Chem. Int. Ed. 2016, 55, 2810–2814.

      Abstract | PDF | Supporting Information



59. Nickel-Catalysed Suzuki–Miyaura Coupling of Amides.

      Nicholas A. Weires, Emma L. Baker and Neil K. Garg. Nat. Chem. 2016, 8, 75–79.

      Abstract | PDF | Supporting Information | C&E News | C&E News Top Research of 2015



58. Discovery of Unclustered Fungal Indole Diterpene Biosynthetic Pathways through Combinatorial Pathway Reassembly in Engineered Yeast.

      Man-Cheng Tang, Hsiao-Ching Lin, Dehai Li, Yi Zou, Jian Li, Wei Xu, Ralph A. Cacho, Maureen E. Hillenmeyer, Neil K. Garg, and Yi Tang.

      J. Am. Chem. Soc. 2015, 137, 13724–13727.

      Abstract | PDF | Supporting Information



  1. 57.Conversion of Amides to Esters by the Nickel-Catalysed Activation of Amide C–N Bonds.
    Liana Hie, Noah F. Fine Nathel, Tejas K. Shah, Emma L. Baker, Xin Hong, Yun-Fang Yang, Peng Liu, K. N. Houk, and Neil K. Garg.
    Nature 2015, 524, 79–83. 

      Abstract | PDF | Supporting Information | C&E News | Nat. Chem. Highlight | Angew. Chem. Int. Ed. Highlight | Synform | C&E News Top

      Research of 2015 | Org. Chem. Highlights


  1. 56.Fischer Indolizations as a Strategic Platform for the Total Synthesis of Picrinine.
    Joel M. Smith, Jesus Moreno, Ben W Boal, and Neil K. Garg. J. Org. Chem. 2015, 80, 8954–8967. (Featured Article)
    Abstract | PDF | Supporting Information
































  1. 55.Generation and Regioselective Trapping of a 3,4-Piperidyne for the Synthesis of Functionalized Heterocycles.
    Travis C. McMahon, Jose M. Medina, Yun-Fang Yang, Bryan J. Simmons, K. N. Houk, and Neil K. Garg.
    J. Am. Chem. Soc. 2015, 137, 4082–4085.
    Abstract | PDF | Supporting Information | JACS Spotlight | C&E News



  1. 54.Elucidation of the Concise Biosynthetic Pathway of the Communesin Indole Alkaloids.
    Hsiao-Ching Lin, Grace Chiou, Yit-Heng Chooi, Travis C. McMahon, Wei Xu, Neil K. Garg, and Yi Tang.
    Angew. Chem. Int. Ed. 2015, 54, 3004–3007. (Selected as a Very Important Paper)
    Abstract | PDF



  1. 53.Computational Predictions of Substituted Benzyne and Indolyne Regioselectivities.
    Elias Picazo, K. N. Houk, and Neil K. Garg. Tetrahedron Lett. 2015, 56, 3511–3514. (Special issue for Professor Harry Wasserman)

      Abstract | PDF



  1. 52.Synthetic Chemistry Fuels Interdisciplinary Approaches to the Production of Artemisinin.
    Michael A. Corsello, and Neil K. Garg. Nat. Prod. Rep. 2015, 32, 359–366.

      Abstract | PDF



  1. 51.Pyridynes and Indolynes as Building Blocks for Functionalized Heterocycles and Natural Products.
    Adam E. Goetz, Tejas K. Shah and Neil K. Garg. Chem. Commun. 2015, 51, 34–45. (Featured Article)
    Abstract | PDF



  1. 50.The Role of Aryne Distortions, Steric Effects, and Charges on Regioselectivities in Aryne Reactions.
    Jose M. Medina, Joel L. Mackey, Neil K. Garg, and K. N. Houk. J. Am. Chem. Soc. 2014, 136, 15798–15805.
    Abstract | PDF | Supporting Information



  1. 49.Total Synthesis of (–)-N-Methylwelwitindolinone B Isothiocyanate via a Chlorinative Oxabicycle Ring-Opening Strategy.
    Nicholas A. Weires, Evan D. Styduhar, Emma L. Baker, and Neil K. Garg. J. Am. Chem. Soc. 2014, 136, 14710–14713.
    Abstract | PDF | Supporting Information | Synfacts Highlight



  1. 48.Cycloadditions of Cyclohexynes and Cyclopentyne.
    Jose M. Medina, Travis C. McMahon, Gonzalo Jiménez-Osés, K. N. Houk, and Neil K. Garg. J. Am. Chem. Soc. 2014, 136, 14706–14709.

       Abstract | PDF | Supporting Information

      



  1. 47.Cascade Reactions: A Driving Force in Akuammiline Alkaloid Total Synthesis.
    Joel M. Smith, Jesus Moreno, Ben W. Boal, and Neil K. Garg. Angew. Chem. Int. Ed. 2015, 54, 400–412.
    Abstract | PDF



  1. 46.Nickel-Catalyzed Amination of Aryl Chlorides and Sulfamates in 2-Methyl-THF
    Noah F. Fine Nathel, Junyong Kim, Liana Hie, Xingyu Jiang, and Neil K. Garg. ACS Catal. 2014, 4, 3289–3293.
    Abstract | PDF | Supporting Information | C&E News



  1. 45.Nickel-Catalyzed Suzuki–Miyaura Cross-Coupling in a Green Alcohol Solvent for an Undergraduate Organic Chemistry Laboratory.
    Liana Hie, Jonah J. Chang, and Neil K. Garg. J. Chem. Educ. 2015, 92, 571–574.  
    Abstract | PDF | Supporting Information


      

  1. 44.Total Synthesis of the Akuammiline Alkaloid Picrinine.
    Joel M. Smith, Jesus Moreno, Ben W. Boal, and Neil K. Garg. J. Am. Chem. Soc. 2014, 136, 4504–4507.
    Abstract | PDF | Supporting Information | Synfacts Highlight



  1. 43.Concise Enantiospecific Total Synthesis of Tubingensin A.
    Adam E. Goetz, Amanda L. Silberstein, Michael A. Corsello, and Neil K. Garg. J. Am. Chem. Soc. 2014, 136, 3036–3039.
    Abstract | PDF | Supporting Information | Synfacts Highlight | Organic Chemistry Portal



  1. 42.Total Syntheses of Indolactam Alkaloids (–)-Indolactam V, (–)-Pendolmycin, (–)-Lyngbyatoxin A, and (–)-Teleocidin A-2.
    Noah F. Fine Nathel, Tejas K. Shah, Sarah M. Bronner, and Neil. K. Garg. Chem. Sci. 2014, 5, 2184–2190.
    Abstract | PDF | Supporting Information



  1. 41.Enabling the Use of Heterocyclic Arynes in Chemical Synthesis.
    Adam E. Goetz and Neil K. Garg. J. Org. Chem. 2014, 79, 846–851.
    Abstract | PDF



  1. 40.Palladium-Catalyzed Acetylation of Arenes.
    Stephen D. Ramgren
    and Neil K. Garg. Org. Lett. 2014, 16, 824–827.
    Abstract | PDF | Supporting Information | C&E News | Organic Chemistry Portal



  1. 39.Enantiospecific Total Synthesis of N-Methylwelwitindolinone D Isonitrile.
    Evan D. Styduhar, Alexander D. Huters, Nicholas A.
    Weires, and Neil K. Garg. Angew. Chem. Int. Ed. 2013, 52, 12422–12425.
    Abstract | PDF | Supporting Information | Synfacts Highlight



  1. 38.Nickel-Catalyzed Suzuki-Miyaura Coupling in Green Solvents.
    Stephen D. Ramgren, Liana Hie, Yuxuan Ye, and Neil K. Garg. Org. Lett. 2013, 15, 3950–3953.
    Abstract | PDF | Supporting Information | Nexus Newsletters



  1. 37.Expanding the Structural Diversity of Polyketides by Exploring the Cofactor Tolerance of an Inline Methyltransferase Domain.
    Jaclyn M. Winter, Grace Chiou, Ian R. Bothwell,, Wei Xu, Neil K. Garg, Minkui Luo, and Yi Tang. Org. Lett. 2013, 15, 3774–3777.
    Abstract | PDF | Supporting Information




  1. 36.EcdGHK are Three Tailoring Iron Oxygenases for Amino Acid Building Blocks of the Echinocandin Scaffold.
    Wei Jiang, Ralph A. Cacho, Grace Chiou, Neil K. Garg, Yi Tang, and Christopher T. Walsh. J. Am. Chem. Soc. 2013, 135, 4457–4466.
    Abstract | PDF | Supporting Information





  1. 35.Synthesis of Diphenylhexatriene by the Pd-Catalyzed Dimerization of Cinnamyl Acetate.
    Tehetena Mesganaw, G.-Yoon J. Im, and Neil K. Garg. J. Org. Chem. 2013, 78, 3391–3393.
    Abstract | PDF | Supporting Information



  1. 34.Regioselective Reactions of 3,4-Pyridynes Enabled by the Aryne Distortion Model.
    Adam E. Goetz and Neil K. Garg. Nat. Chem. 2013, 5, 54–60.
    Abstract | PDF | Supporting Information | Synfacts Highlight




  1. 33.Ni- and Fe-Catalyzed Cross-Coupling Reactions of Phenol Derivatives.
    Tehetena Mesganaw and Neil K. Garg. Org. Process Res. Dev. 2013, 17, 29–39.
    Abstract | PDF


  1. 32.Identification and Characterization of the Chaetoviridin and Chaetomugilin Gene Cluster in Chaetomium globosum Reveal Dual Functions of an Iterative Highly-Reducing Polyketide Synthase.
    Jaclyn M. Winter, Michio Sato, Satoru Sugimoto, Grace Chiou, Neil K. Garg, Yi Tang, and Kenji Watanabe.
    J. Am. Chem. Soc. 2012, 134, 17900–17903.
    Abstract | PDF | Supporting Information



  1. 31.Interrupted Fischer Indolization Approach toward the Communesin Alkaloids and Perophoramidine.
    Alex W. Schammel, Grace Chiou, and Neil K. Garg. Org. Lett. 2012, 14, 4556–4559.
    Abstract | PDF | Supporting Information



  1. 30.Steric Effects Compete with Aryne Distortion to Control Regioselectivities of Nucleophilic Additions to 3-Silylarynes.
    Sarah M. Bronner, Joel L. Mackey, K. N. Houk, and Neil K. Garg. J. Am. Chem. Soc. 2012, 134, 13966–13969.
    Abstract | PDF | Supporting Information



  1. 29.Nickel-Catalyzed Amination of Aryl Sulfamates and Carbamates Using an Air-Stable Precatalyst.
    Liana Hie, Stephen D. Ramgren, Tehetena Mesganaw, and Neil K. Garg. Org. Lett. 2012, 14, 4182–4185.
    Abstract | PDF | Supporting Information



  1. 28.Iron-Catalyzed Alkylations of Aryl Sulfamates and Carbamates.
    Amanda L. Silberstein, Stephen D. Ramgren, and Neil K. Garg. Org. Lett. 2012, 14, 3796–3799.
    Abstract | PDF | Supporting Information | Synfacts Highlight | Organic Chemistry Portal



  1. 27.Cine Substitution of Arenes Using the Aryl Carbamate as a Removable Directing Group.
    Tehetena Mesganaw, Noah F. Fine Nathel, and Neil K. Garg. Org. Lett. 2012, 14, 2918–2921.
    Abstract | PDF | Supporting Information



  1. 26.Total Syntheses of the Elusive Welwitindolinones with Bicyclo[4.3.1]cores.
    Alexander D. Huters, Evan D. Styduhar, and Neil K. Garg. Angew. Chem. Int. Ed. 2012, 51, 3758–3765.
    Abstract | PDF



  1. 25.An Efficient Computational Model to Predict the Synthetic Utility of Heterocyclic Arynes.
    Adam E. Goetz, Sarah M. Bronner, Jordan D. Cisneros, Joshua M. Melamed, Robert S. Paton, K. N. Houk, and Neil K. Garg.
    Angew. Chem. Int. Ed. 2012, 51, 2758–2762.
    Abstract | PDF | Supporting Information



  1. 24.Total Synthesis of Oxidized Welwitindolinones and (–)-N-Methylwelwitindolinone C Isonitrile.
    Kyle W. Quasdorf, Alexander D. Huters, Michael W. Lodewyk, Dean J. Tantillo, and Neil K. Garg. J. Am. Chem. Soc. 2012, 134, 1396–1399.
    Abstract | PDF | Supporting Information



  1. 23.Synthesis of (+)-Phenserine using an Interrupted Fischer Indolization Reaction.
    Alex W. Schammel, Grace Chiou, Neil K. Garg. J. Org. Chem. 2012, 77, 725–728.
    Abstract | PDF | Supporting Information



  1. 22.Total Synthesis of (–)-N-Methylwelwitindolinone C Isothiocyanate.
    Alexander D. Huters, Kyle W. Quasdorf, Evan D. Styduhar, and Neil K. Garg. J. Am. Chem. Soc. 2011, 133, 15797–15799.
    Abstract | PDF | Supporting Information | C&E News Highlight | Synfacts Highlight | Nature Chemistry | Organic Chemistry Portal
































  1. 21.Understanding and Modulating Indolyne Regioselectivities.
    Sarah M. Bronner, Adam E. Goetz, and Neil K. Garg. Synlett 2011, 18, 2599–2604. (invited SYNPACTS article)
    Abstract | PDF



  1. 20.Nickel-Catalyzed Amination of Aryl Carbamates and Sequential Site-Selective Cross-Couplings.
    Tehetena Mesganaw, Amanda L. Silberstein, Stephen D. Ramgren, Noah F. Fine Nathel, Xin Hong, Peng Liu, and Neil K. Garg.
    Chem. Sci. 2011, 2, 1766–1771.
    Abstract | PDF | Supporting Information



  1. 19.Total Synthesis of (±)-Aspidophylline A.
    Liansuo Zu, Ben W. Boal, and Neil K. Garg. J. Am. Chem. Soc. 2011, 133, 8877–8879.
    Abstract | PDF | Supporting Information | Synfacts Highlight | Org. Highlights



  1. 18.Suzuki–Miyaura Cross-Coupling of Aryl Carbamates and Sulfamates: Experimental and Computational Studies.
    Kyle W. Quasdorf, Aurora Antoft-Finch, Peng Liu, Amanda L. Silberstein, Anna Komaromi, Tom Blackburn, Stephen D. Ramgren, K. N. Houk, Victor Snieckus, and Neil K. Garg.
    J. Am. Chem. Soc. 2011, 133, 6352–6363.
    Abstract | PDF | Supporting Information | Synfacts Highlight



  1. 17.Why Do Some Fischer Indolizations Fail?
    Nihan Çelebi-Olcüm, Ben W. Boal, Alexander D. Huters, Neil K. Garg, and K. N. Houk. J. Am. Chem. Soc. 2011, 133, 5752–5755.
    Abstract | PDF | Supporting Information



  1. 16.Overturning Indolyne Regioselectivities and Synthesis of Indolactam V.
    Sarah M. Bronner, Adam E. Goetz, and Neil K. Garg. J. Am. Chem. Soc. 2011, 133, 3832–3835.
    Abstract | PDF | Supporting Information | Synpacts Highlight



  1. 15.A Fungal Nonribosomal Peptide Synthetase Module that can Synthesize Thiopyrazines.
    Kangjian Qiao, Hui Zhou, Wei Xu, Wenjun Zhang, Neil K. Garg, and Yi Tang. Org. Lett. 2011, 13, 1758–1761.
    Abstract | PDF | Supporting Information





  1. 14.Nickel-Catalyzed Amination of Aryl Sulfamates.
    Stephen D. Ramgren, Amanda L. Silberstein, Yang Yang, and Neil K. Garg. Angew. Chem. Int. Ed. 2011, 50, 2171–2173.
    Abstract | PDF | Supporting Information | Synfacts Highlight



  1. 13.Nickel-Catalyzed Cross-Couplings Involving Carbon–Oxygen Bonds.
    Brad M. Rosen, Kyle W. Quasdorf, Daniella A. Wilson, Na Zhang, Ana-Maria Resmerita, Neil K. Garg, and Virgil Percec.
    Chem. Rev. 2011, 111, 1346–1416 (invited contribution).
    Abstract | PDF


  1. 12.Indoles and Indolizidines in Heterocycles in Natural Product Synthesis.
    Sarah M. Bronner, G-Yoon J. Im, and Neil K. Garg; K. C. Majumdar and S. K. Chattopadhyay, Eds.; Wiley–VCH, 2011.


  1. 11.Indolyne Experimental and Computational Studies: Synthetic Applications and Origins of Selectivities of Nucleophilic Additions.
    G-Yoon J. Im, Sarah M. Bronner, Adam E. Goetz, Robert S. Paton, Paul H.-Y. Cheong, K. N. Houk, and Neil K. Garg.
    J. Am. Chem. Soc. 2010, 132, 17933–17944.
    Abstract | PDF | Supporting Information



  1. 10.Bis(tricyclohexylphosphine)dichloronickel.
    Kyle W. Quasdorf and Neil K. Garg. Encyclopedia of Reagents for Organic Synthesis, 2010 (invited contribution).
    Link | PDF



  1. 9.Synthetic Studies Inspired by Vinigrol.
    Alexander D. Huters and Neil K. Garg. Chem. Eur. J. 2010, 16, 8586–8595.

   Abstract | PDF



  1. 8.Exploration of the Interrupted Fischer Indolization Reaction.
    Alex W. Schammel, Ben W. Boal, Liansuo Zu, Tehetena Mesganaw, and Neil K. Garg. Tetrahedron 2010, 66, 4687–4695.
    (Special issue for Professor Brian Stoltz’s receipt of the Tetrahedron Young Investigator Award)
    Abstract | PDF | Supporting Information

  


  1. 7.Indolyne and Aryne Distortions and Nucleophilic Regioselectivities.
    Paul H.-Y. Cheong, Robert S. Paton, Sarah M. Bronner, G-Yoon J. Im, Neil K. Garg, and K. N. Houk. J. Am. Chem. Soc. 2010, 132, 1267–1269.
    Abstract | PDF | Supporting Information | Chemistry World Highlight



  1. 6.Suzuki–Miyaura Coupling of Aryl Carbamates, Carbonates, and Sulfamates.
    Kyle W. Quasdorf, Michelle Riener, Krastina V. Petrova, and Neil K. Garg. J. Am. Chem. Soc. 2009, 131, 17748–17749.
    Abstract | PDF | Supporting Information | Synfacts Highlight



  1. 5.Efficient Synthesis of 2-(Trimethylsilyl)phenyl Trifluoromethanesulfonate: A Versatile Precursor to o-Benzyne.
    Sarah M. Bronner and Neil K. Garg. J. Org. Chem. 2009, 74, 8842–8843.
    Abstract | PDF | Supporting Information | ACS Noteworthy Chemistry Highlight



  1. 4.An Interrupted Fischer Indolization Approach Toward Fused Indoline-Containing Natural Products.
    Ben W. Boal, Alex W. Schammel, and Neil K. Garg. Org. Lett. 2009, 11, 3458–3461.
    Abstract | PDF | Supporting Information



  1. 3.Concise Synthesis of the Bicyclic Scaffold of N-Methylwelwitindolinone C Isothiocyanate via an Indolyne Cyclization.
    Xia Tian, Alexander D. Huters, Colin J. Douglas, and Neil K. Garg. Org. Lett. 2009, 11, 2349–2351.
    Abstract | PDF | Supporting Information



  1. 2.Indolynes as Electrophilic Indole Surrogates: Fundamental Reactivity and Synthetic Applications.
    Sarah M. Bronner, Kevin B. Bahnck, and Neil K. Garg. Org. Lett. 2009, 11, 1007–1010.
    Abstract | PDF | Supporting Information



  1. 1.Cross-Coupling Reactions of Aryl Pivalates with Boronic Acids.
    Kyle W. Quasdorf, Xia Tian, and Neil K. Garg. J. Am. Chem. Soc. 2008, 130, 14422–14423.
    Abstract | PDF | Supporting Information | Synfacts Highlight




Patents


2. Amination of Aryl Alcohol Derivatives. Neil K. Garg, Stephen D. Ramgren, Amanda L. Silberstein, and Kyle W. Quasdorf. U.S. Provisional      
    Patent Application, filed January, 2011.


1. Cross-Coupling of Phenolic Derivatives. Neil K. Garg, Kyle W. Quasdorf, and Xia Tian. U.S. Patent Application, filed September, 2010.

 

Publications (Research Contributions)

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