Selected References

Weilin Chen, Martin Diaz, Juston Rockwell, Carolyn B. Knobler and M. Frederick Hawthorne, "Synthesis and Characterization of Water-Soluble Boron-Substituted Ortho-Carborane Derivatives," Comptes Rendus de l'Académie des Sciences - Série IIc - Chemie, 3, 223 (2000).

M. Frederick Hawthorne and Andreas Maderna, "Applications of Radiolabeled Boron Clusters to the Diagnosis and Treatment of Cancer," Chem. Rev., 99, 3421 (1999).

Akira Nakanishi, Lufeng Guan, Robert R. Kane, Harumi Kasamatsu and M. Frederick Hawthorne, "Toward a Cancer Therapy with Boron-rich Oligomeric Phosphate Diesters that Target the Cell Nucleus," Proc. Natl. Acad. Sci. USA, 96, 238, (1999).

M. Frederick Hawthorne, "New Horizons for Therapy Based on the Boron Neutron Capture Reaction," Mol. Med. Today , 4, No. 4, 174 (1998).

Rachel A. Watson-Clark, Mona Lisa Banquerigo, Kenneth Shelly, M. Frederick Hawthorne and Ernest L. Brahn, "Model Studies Directed Toward the Application of Boron Neutron Capture Therapy to Rheumatoid Arthritis: Boron Delivery by Liposomes to Rat Collagen-Induced Arthritis," Proc. Natl. Acad. Sci. USA, 95, 2531 (1998).

Lufeng Guan, Letitia A. Wims, Robert R. Kane, Mark Smuckler, Sherie L. Morrison and M. Frederick Hawthorne, "Homogeneous Immunoconjugates for Boron Neutron Capture Therapy: Design, Synthesis and Preliminary Characterization," Proc. Natl. Acad. Sci. USA, 95, 13206, (1998).

Charng-Jui Chen, Robert R. Kane, F. James Primus, Gyórgy Szalai, M. Frederick Hawthorne and John E. Shively, "Synthesis and Characterization of Oligomeric Nido-carboranyl Phosphate Diester Conjugates to Antibody and Antibody Fragments for Potential Use in Boron Neutron Capture Therapy of Solid Tumors," Bioconjugate Chem., 5, 557, (1994).

Robert R. Kane, Karin Drechsel and M. Frederick Hawthorne, "Automated Syntheses of Carborane-Derived Homogeneous Oligophosphates: Reagents for Use in the Immunoprotein-Mediated Boron Neutron Capture Therapy (BNCT) of Cancer," J. Am. Chem. Soc., 115, 8853 (1993).

Robert R. Kane, Christine S. Lee, Karin Drechsel, and M. Frederick Hawthorne, "Solution-Phase Synthesis of Boron-Rich Phosphates," J. Org. Chem., 58, 3227, (1993).

Raymond J. Paxton, Barbara G. Beatty, M. Frederick Hawthorne, Aravamuthan Varadarajan, Lawrence E. Williams, Frederick L. Curtis, Carolyn B. Knobler, J. David Beatty and John E. Shively, "A Transition Metal Complex (Venus Flytrap Cluster) for Radioimmunodetection and Radioimmunotherapy," Proc. Natl. Acad. Sci., 88, 3387 (1991).

M. Frederick Hawthorne, Aravamuthan Varadarajan, Carolyn B. Knobler, Sarmistha Chakrabarti, Raymond J. Paxton, Barbara G. Beatty and Frederick L. Curtis, "Radiometallacarboranes as Tumor Imaging Reagents," J. Am. Chem. Soc., 112, 5365 (1990).

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